CompChem-Database: details for selected entry

ChEBI185963 (100536)

FormulaC27H38O
MW378.6
InChIKeyAJRNPFZYKICTEM-UHFFFAOYNA-N
Entry_Date2023-11-01
Net_Charge0
Number_Atoms66
Number_Heavy_Atoms28
Number_Rings4
Number_Bonds69
Rotat_Bonds4
Unbranched_Chain3
Chiral_Centers5
ONatoms1
HB_Donor0
HB_Acceptor1
OpenEye_HB_Donors0
OpenEye_HB_Acceptors1
Lipinski_HB_Donors0
Lipinski_HB_Acceptors1
Lipinski_Violations1
XLogP30
XLogP6.04
logP7.2131
PSA17.07
MR121.231
ABS0.55
Solubilitypoorly
AggregatorPass
PM7_Heat_of_Formation_kcal_per_mol-48.31988
PM7_Total_Energy_ev-4125.1808
PM7_Electronic_Energy_ev-39268.50948
PM7_Dipole_Debye6.33626
PM7_Point_GroupC1
PM7_HOMO_Energy_ev-8.763
PM7_LUMO_Energy_ev-0.666
PM7_COSMO_Area_square_ang418.76
PM7_COSMO_Volue_cubic_ang522.36
PM7_Electron_Affinity_ev0.666
PM7_Ionization_Energy_ev8.763
PM7_Energy_Gap_ev8.097
PM7_Global_Hardness_ev4.0485
PM7_Global_Softness_ev0.24700506360380386
PM7_Chemical_Potential_ev-4.7145
PM7_Electronigativity_ev4.7145
PM7_Back_Donation_Energy_ev-1.012125
PM7_Electrophilicity_ev2.7450302889959244
OPENEYE_Name(9~{R},10~{R},13~{R},17~{R})-17-[(~{E},1~{R})-1,5-dimethylhex-2-enyl]-10,13-dimethyl-1,2,9,11,12,15,16,17-octahydrocyclopenta[a]phenanthren-3-one
SMILESC1=CC2=C3CCC(C3(CCC2C4(C1=CC(=O)CC4)C)C)C(C=CCC(C)C)C
Canonical_SMILESCC(C/C=C/[C@H]([C@H]1CCC2=C3[C@H](CC[C@]12C)[C@@]1(C)CCC(=O)C=C1C=C3)C)C
InChI1/C27H38O/c1-18(2)7-6-8-19(3)23-11-12-24-22-10-9-20-17-21(28)13-15-26(20,4)25(22)14-16-27(23,24)5/h6,8-10,17-19,23,25H,7,11-16H2,1-5H3
InChI_3D1S/C27H38O/c1-18(2)7-6-8-19(3)23-11-12-24-22-10-9-20-17-21(28)13-15-26(20,4)25(22)14-16-27(23,24)5/h6,8-10,17-19,23,25H,7,11-16H2,1-5H3/b8-6+/t19-,23-,25+,26+,27-/m1/s1
AuxInfo1/0/N:23,24,22,20,21,8,25,9,1,2,12,10,11,14,13,15,3,27,26,4,7,5,17,6,16,18,19,28/E:(1,2)/rA:66cCCCCCCCCCCCCCCCCCCCCCCCCCCCOHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHH/rB:d1;;s1d3;s2;d5;s3;;w8;s6;s7;s10;s11;;s14;s5s14;s12;s4s13s16;s6s15s17;s18;s19;;;;s8;s9s17s22;s23s24s25;d7;s1;s2;s3;s8;s9;s10;s10;s11;s11;s12;s12;s13;s13;s14;s14;s15;s15;s16;s17;s20;s20;s20;s21;s21;s21;s22;s22;s22;s23;s23;s23;s24;s24;s24;s25;s25;s26;s27;/rC:2.6037,-.4989,0;3.4748,.0023,0;.8679,-.4977,0;1.7371,0,0;3.4759,1.0071,0;4.3477,1.5084,0;;4.6796,5.9949,0;4.8555,5.0105,0;6.0915,1.5061,0;0,1.0056,0;6.0928,2.5162,0;.8679,1.5135,0;2.5967,2.5196,0;3.4743,3.0237,0;2.6012,1.5123,0;5.2187,3.0279,0;1.7358,1.0056,0;4.349,2.5184,0;.8686,.5076,0;5.2163,2.0206,0;3.4464,5.1306,0;6.8533,6.5192,0;6.9735,7.9283,0;5.4442,6.6394,0;4.0908,4.366,0;6.2089,7.2839,0;-.8653,-.5013,0;2.6036,-.9989,0;3.9075,-.2483,0;.8677,-.9977,0;4.2094,6.1649,0;5.3257,4.8405,0;6.5915,1.5055,0;6.0908,1.0061,0;-.4922,.9178,0;-.1728,1.4748,0;6.2659,2.9853,0;6.585,2.428,0;.5458,1.8959,0;1.19,1.8959,0;2.1045,2.4317,0;2.4257,2.9894,0;3.1535,3.4072,0;3.796,3.4064,0;2.6027,1.0123,0;5.5408,3.4103,0;1.1176,.074,0;.6196,.9412,0;.435,.2586,0;5.4652,2.4542,0;4.9674,1.5869,0;5.6499,1.7717,0;3.0641,4.8083,0;3.8287,5.4528,0;3.1241,5.5129,0;6.471,6.197,0;7.2357,6.8415,0;7.1756,6.1369,0;7.2957,7.546,0;6.6512,8.3107,0;7.3558,8.2506,0;5.7665,6.2571,0;5.122,7.0217,0;3.7085,4.0437,0;5.8866,7.6662,0;
DuplicatesChEBI185963
mol2_Path/CCDB/ChEBI/Database/Compound-0000150000-0000199999/Compound-0000185750-0000185999/ChEBI185963.mol2
pdbqt_Path/CCDB/ChEBI/Database/Compound-0000150000-0000199999/Compound-0000185750-0000185999/ChEBI185963.pdbqt
sdf_Path/CCDB/ChEBI/Database/Compound-0000150000-0000199999/Compound-0000185750-0000185999/ChEBI185963.sdf