CompChem-Database: details for selected entry

CHEMBL5193803_p0_t1 (2536349)

FormulaC21H24N3O3
MW366.44
InChIKeyFLCSMUCKUNAXHO-QYLZYXQNNA-O
Entry_Date2023-09-01
Net_Charge1
Number_Atoms51
Number_Heavy_Atoms27
Number_Rings3
Number_Bonds53
Rotat_Bonds8
Unbranched_Chain5
Chiral_Centers0
ONatoms6
HB_Donor1
HB_Acceptor1
OpenEye_HB_Donors2
OpenEye_HB_Acceptors1
Lipinski_HB_Donors2
Lipinski_HB_Acceptors6
Lipinski_Violations0
XLogP30
XLogP4.37
logP3.6537
PSA83.77
MR114.74
ABS0.55
Solubilityhighly
AggregatorPass
PM7_Heat_of_Formation_kcal_per_mol136.69188
PM7_Total_Energy_ev-4338.91415
PM7_Electronic_Energy_ev-34251.60535
PM7_Dipole_Debye12.46627
PM7_Point_GroupC1
PM7_HOMO_Energy_ev-11.012
PM7_LUMO_Energy_ev-6.199
PM7_COSMO_Area_square_ang407.84
PM7_COSMO_Volue_cubic_ang450.48
PM7_Electron_Affinity_ev6.199
PM7_Ionization_Energy_ev11.012
PM7_Energy_Gap_ev4.813
PM7_Global_Hardness_ev2.4065
PM7_Global_Softness_ev0.415541242468315
PM7_Chemical_Potential_ev-8.6055
PM7_Electronigativity_ev8.6055
PM7_Back_Donation_Energy_ev-0.601625
PM7_Electrophilicity_ev15.386376532308331
OPENEYE_Name(~{Z})-[4-[(4-butoxy-3-methoxy-phenyl)methyl]-5-oxo-imidazol-2-ylidene]-phenyl-ammonium
SMILESc1ccc(cc1)[NH+]=C2N=C(C(=O)N2)Cc3ccc(c(c3)OC)OCCCC
Canonical_SMILESCCCCOc1ccc(cc1OC)CC1=N/C(=[NH]c2ccccc2)/NC1=O
InChI1/C21H23N3O3/c1-3-4-12-27-18-11-10-15(14-19(18)26-2)13-17-20(25)24-21(23-17)22-16-8-6-5-7-9-16/h5-11,14H,3-4,12-13H2,1-2H3,(H,22,24,25)/p+1/fC21H24N3O3/h22,24H/q+1
InChI_3D1S/C21H24N3O3/c1-3-4-12-27-18-11-10-15(14-19(18)26-2)13-17-20(25)24-21(23-17)22-16-8-6-5-7-9-16/h5-11,14,22H,3-4,12-13H2,1-2H3,(H,24,25)/b22-21+
AuxInfo1/1/N:16,17,19,20,1,2,3,5,6,4,7,21,18,8,9,10,13,11,12,14,15,24,22,23,25,26,27/E:(6,7)(8,9)/F:m/E:m/rA:51nCCCCCCCCCCCCCCCCCCCCCNNN+OOOHHHHHHHHHHHHHHHHHHHHHHHH/rB:d1;s1;;s2;d3;d4;;s4d8;d5s6;s7;s8d11;;s13;;;;s9s13;s16;s19;s20;d13s15;s14s15;s10w15;d14;s12s17;s11s21;s1;s2;s3;s4;s5;s6;s7;s8;s16;s16;s16;s17;s17;s17;s18;s18;s19;s19;s20;s20;s21;s21;s23;s24;/rC:4.4991,-.7577,0;3.5485,-1.0682,0;4.7111,.2196,0;-.7735,-2.5312,0;2.8023,-.3946,0;3.965,.8932,0;-1.3589,-3.342,0;-2.1774,-1.5115,0;-1.1777,-1.6165,0;3.0068,.5895,0;-2.3586,-3.237,0;-2.7729,-2.3213,0;;-.3065,.9519,0;1.3131,.9519,0;-1.3057,-7.697,0;-4.3551,-3.026,0;-.5889,-.8082,0;-1.7152,-6.7847,0;-2.1248,-5.8724,0;-2.5343,-4.9602,0;1.0014,0,0;.5007,1.5426,0;2.2646,1.2597,0;-1.2577,1.2606,0;-3.7675,-2.2169,0;-2.9439,-4.0479,0;4.8702,-1.0927,0;3.4446,-1.5573,0;5.1871,.3728,0;-.2762,-2.5834,0;2.3271,-.5499,0;4.071,1.3819,0;-1.1548,-3.7984,0;-2.3795,-1.0542,0;-1.7618,-7.9018,0;-.8495,-7.4923,0;-1.1009,-8.1532,0;-3.9506,-3.3198,0;-4.7597,-2.7321,0;-4.649,-3.4305,0;-.1847,-1.1027,0;-.993,-.5138,0;-1.2591,-6.58,0;-2.1714,-6.9895,0;-1.6686,-5.6677,0;-2.5809,-6.0772,0;-2.9905,-5.1649,0;-2.0782,-4.7554,0;.4999,2.0426,0;2.3692,1.7486,0;
DuplicatesCHEMBL5193803_p0_t1;CHEMBL5193803_p7_t1
mol2_Path/CCDB/ChEMBL/Database/Compound-0005150000-0005199999/Compound-0005193750-0005193999/CHEMBL5193803_p0_t1.mol2
pdbqt_Path/CCDB/ChEMBL/Database/Compound-0005150000-0005199999/Compound-0005193750-0005193999/CHEMBL5193803_p0_t1.pdbqt
sdf_Path/CCDB/ChEMBL/Database/Compound-0005150000-0005199999/Compound-0005193750-0005193999/CHEMBL5193803_p0_t1.sdf