CompChem-Database: details for selected entry

CHEMBL103075_m2_s0 (3177)

FormulaC19H29NO7P
MW414.41
InChIKeySGHLYPWBEXWOJR-KNAGUMQPNA-K
Entry_Date2023-09-01
Net_Charge-3
Number_Atoms60
Number_Heavy_Atoms28
Number_Rings0
Number_Bonds59
Rotat_Bonds17
Unbranched_Chain3
Chiral_Centers1
ONatoms8
HB_Donor4
HB_Acceptor6
OpenEye_HB_Donors1
OpenEye_HB_Acceptors6
Lipinski_HB_Donors1
Lipinski_HB_Acceptors8
Lipinski_Violations0
XLogP30
XLogP-0.25
logP3.7228
PSA142.97
MR108.871
ABS0.56
Solubilitypoorly
AggregatorPass
PM7_Heat_of_Formation_kcal_per_mol-292.55757
PM7_Total_Energy_ev-5154.34707
PM7_Electronic_Energy_ev-43762.43866
PM7_Dipole_Debye27.86924
PM7_Point_GroupC1
PM7_HOMO_Energy_ev1.948
PM7_LUMO_Energy_ev8.059
PM7_COSMO_Area_square_ang396.56
PM7_COSMO_Volue_cubic_ang516.86
PM7_Electron_Affinity_ev-8.059
PM7_Ionization_Energy_ev-1.948
PM7_Energy_Gap_ev6.111
PM7_Global_Hardness_ev3.0555
PM7_Global_Softness_ev0.3272786777941417
PM7_Chemical_Potential_ev5.0035
PM7_Electronigativity_ev-5.0035
PM7_Back_Donation_Energy_ev-0.763875
PM7_Electrophilicity_ev4.096712853870071
OPENEYE_Name(2~{S})-3-oxo-2-(phosphonatooxymethyl)-3-[[(2~{E},6~{E})-3,7,11-trimethyldodeca-2,6,10-trienyl]amino]propanoate
SMILESC(=C(C)C)CCC(=CCCC(=CCNC(=O)C(C(=O)[O-])COP(=O)([O-])[O-])C)C
Canonical_SMILESC/C(=CCNC(=O)[C@@H](C(=O)O)COP(=O)(O)O)/CC/C=C(CCC=C(C)C)/C
InChI1/C19H32NO7P/c1-14(2)7-5-8-15(3)9-6-10-16(4)11-12-20-18(21)17(19(22)23)13-27-28(24,25)26/h7,9,11,17H,5-6,8,10,12-13H2,1-4H3,(H,20,21)(H,22,23)(H2,24,25,26)/p-3/fC19H29NO7P/h20H/q-3
InChI_3D1S/C19H32NO7P/c1-14(2)7-5-8-15(3)9-6-10-16(4)11-12-20-18(21)17(19(22)23)13-27-28(24,25)26/h7,9,11,17H,5-6,8,10,12-13H2,1-4H3,(H,20,21)(H,22,23)(H2,24,25,26)/b15-9+,16-11+/t17-/m0/s1
AuxInfo1/1/N:9,10,11,12,13,14,1,16,2,17,3,15,18,4,5,6,19,7,8,20,24,21,25,22,23,26,27,28/E:(1,2)(22,23)(24,25,26)/F:m/E:m/rA:57cCCCCCCCCCCCCCCCCCCCNO-O-O-OOOOPHHHHHHHHHHHHHHHHHHHHHHHHHHHHH/rB:;;d1;w2;w3;;;s4;s4;s5;s6;s1;s2;s3;s5s13;s6s14;;s7s8s18;s7s15;s8;;;d7;d8;;s18;s22s23d26s27;s1;s2;s3;s9;s9;s9;s10;s10;s10;s11;s11;s11;s12;s12;s12;s13;s13;s14;s14;s15;s15;s16;s16;s17;s17;s18;s18;s19;s20;/rC:;-1,3.4641,0;2.5,4.3301,0;-.5,-.866,0;-1.5,2.5981,0;2,3.4641,0;.5,6.0622,0;-.5,7.7942,0;0,-1.7321,0;-1.5,-.866,0;-2.5,2.5981,0;2.5,2.5981,0;-.5,.866,0;0,3.4641,0;2,5.1962,0;-1,1.7321,0;1,3.4641,0;-.866,6.4282,0;0,6.9282,0;1.5,6.0622,0;-1.5,7.7942,0;-3.4641,4.9282,0;-3.0981,6.2942,0;0,5.1962,0;0,8.6603,0;-2.0981,4.5622,0;-1.7321,5.9282,0;-2.5981,5.4282,0;.5,0,0;-1.25,3.8971,0;3,4.3301,0;-.433,-1.9821,0;.433,-1.4821,0;.25,-2.1651,0;-1.5,-1.366,0;-1.5,-.366,0;-2,-.866,0;-2.5,3.0981,0;-2.5,2.0981,0;-3,2.5981,0;2.933,2.8481,0;2.067,2.3481,0;2.75,2.1651,0;-.067,1.116,0;-.933,.616,0;0,3.9641,0;0,2.9641,0;1.567,4.9462,0;2.433,5.4462,0;-1.433,1.4821,0;-.567,1.9821,0;1,2.9641,0;1,3.9641,0;-.616,5.9952,0;-1.116,6.8612,0;.433,7.1782,0;1.75,6.4952,0;
DuplicatesCHEMBL103075_m2_s0
mol2_Path/CCDB/ChEMBL/Database/Compound-0000100000-0000149999/Compound-0000103000-0000103249/CHEMBL103075_m2_s0.mol2
pdbqt_Path/CCDB/ChEMBL/Database/Compound-0000100000-0000149999/Compound-0000103000-0000103249/CHEMBL103075_m2_s0.pdbqt
sdf_Path/CCDB/ChEMBL/Database/Compound-0000100000-0000149999/Compound-0000103000-0000103249/CHEMBL103075_m2_s0.sdf