CompChem-Database: details for selected entry

CHEMBL103162 (3272)

FormulaC20H32N2O3
MW348.48
InChIKeyOARLMKKFYRMEGT-XBTAAFKLNA-N
Entry_Date2023-09-01
Net_Charge0
Number_Atoms57
Number_Heavy_Atoms25
Number_Rings1
Number_Bonds57
Rotat_Bonds16
Unbranched_Chain11
Chiral_Centers0
ONatoms5
HB_Donor2
HB_Acceptor2
OpenEye_HB_Donors2
OpenEye_HB_Acceptors2
Lipinski_HB_Donors2
Lipinski_HB_Acceptors5
Lipinski_Violations1
XLogP30
XLogP5.03
logP4.9515
PSA67.43
MR101.376
ABS0.55
Solubilityvery
AggregatorPass
PM7_Heat_of_Formation_kcal_per_mol-158.94077
PM7_Total_Energy_ev-4148.49235
PM7_Electronic_Energy_ev-35282.70191
PM7_Dipole_Debye2.84058
PM7_Point_GroupC1
PM7_HOMO_Energy_ev-9.63
PM7_LUMO_Energy_ev-0.125
PM7_COSMO_Area_square_ang382.58
PM7_COSMO_Volue_cubic_ang481.82
PM7_Electron_Affinity_ev0.125
PM7_Ionization_Energy_ev9.63
PM7_Energy_Gap_ev9.505
PM7_Global_Hardness_ev4.7525
PM7_Global_Softness_ev0.21041557075223566
PM7_Chemical_Potential_ev-4.8775
PM7_Electronigativity_ev4.8775
PM7_Back_Donation_Energy_ev-1.188125
PM7_Electrophilicity_ev2.502893871646502
OPENEYE_Namebenzyl ~{N}-[2-(decylamino)-2-oxo-ethyl]carbamate
SMILESc1ccc(cc1)COC(=O)NCC(=O)NCCCCCCCCCC
Canonical_SMILESCCCCCCCCCCNC(=O)CNC(=O)OCc1ccccc1
InChI1/C20H32N2O3/c1-2-3-4-5-6-7-8-12-15-21-19(23)16-22-20(24)25-17-18-13-10-9-11-14-18/h9-11,13-14H,2-8,12,15-17H2,1H3,(H,21,23)(H,22,24)/f/h21-22H
InChI_3D1S/C20H32N2O3/c1-2-3-4-5-6-7-8-12-15-21-19(23)16-22-20(24)25-17-18-13-10-9-11-14-18/h9-11,13-14H,2-8,12,15-17H2,1H3,(H,21,23)(H,22,24)
AuxInfo1/1/N:9,12,13,14,15,16,17,18,1,2,3,19,4,5,20,11,10,6,7,8,21,22,23,24,25/E:(10,11)(13,14)/F:m/E:m/rA:57nCCCCCCCCCCCCCCCCCCCCNNOOOHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHHH/rB:d1;s1;s2;d3;d4s5;;;;s6;s7;s9;s12;s13;s14;s15;s16;s17;s18;s19;s7s20;s8s11;d7;d8;s8s10;s1;s2;s3;s4;s5;s9;s9;s9;s10;s10;s11;s11;s12;s12;s13;s13;s14;s14;s15;s15;s16;s16;s17;s17;s18;s18;s19;s19;s20;s20;s21;s22;/rC:;-.8675,.4975,0;.8675,.4975,0;-.8675,1.5027,0;.8675,1.5027,0;0,2.0104,0;2.5981,6.5104,0;.866,4.5104,0;12.1244,11.0104,0;0,3.0104,0;1.732,6.0104,0;11.2583,10.5104,0;10.3923,10.0104,0;9.5263,9.5104,0;8.6603,9.0104,0;7.7942,8.5104,0;6.9282,8.0104,0;6.0622,7.5104,0;5.1962,7.0104,0;4.3301,6.5104,0;3.4641,6.0104,0;.866,5.5104,0;2.5981,7.5104,0;1.7321,4.0104,0;0,4.0104,0;0,-.5,0;-1.3001,.2469,0;1.3001,.2469,0;-1.3012,1.7514,0;1.3012,1.7514,0;12.3744,10.5774,0;11.8744,11.4434,0;12.5574,11.2604,0;.5,3.0104,0;-.5,3.0104,0;1.482,6.4434,0;1.982,5.5774,0;11.0083,10.9434,0;11.5083,10.0774,0;10.1423,10.4434,0;10.6423,9.5774,0;9.2763,9.9434,0;9.7763,9.0774,0;8.4103,9.4434,0;8.9103,8.5774,0;7.5442,8.9434,0;8.0442,8.0774,0;6.6782,8.4434,0;7.1782,7.5774,0;5.8122,7.9434,0;6.3122,7.0774,0;4.9462,7.4434,0;5.4462,6.5774,0;4.0801,6.9434,0;4.5801,6.0774,0;3.4641,5.5104,0;.433,5.7604,0;
DuplicatesCHEMBL103162
mol2_Path/CCDB/ChEMBL/Database/Compound-0000100000-0000149999/Compound-0000103000-0000103249/CHEMBL103162.mol2
pdbqt_Path/CCDB/ChEMBL/Database/Compound-0000100000-0000149999/Compound-0000103000-0000103249/CHEMBL103162.pdbqt
sdf_Path/CCDB/ChEMBL/Database/Compound-0000100000-0000149999/Compound-0000103000-0000103249/CHEMBL103162.sdf